circRNA basic information
circBase ID: hsa_circ_0000284
Name: hsa_circ_HIPK3
Synonym: circ_0000284 / circHIPK3
Host Gene: HIPK3
Genomic location(hg19): chr11:33307958-33309057:+
Genomic location(hg38): chr11:33286412-33287511:+
Subcellular localization: cytoplasm
 
 
 
 
 
 
 
Disease basic information
MONDO ID:
0003210
MONDO name: intrahepatic cholangiocarcinoma
Disease details: intrahepatic cholangiocarcinoma / ICC
Disease DO ID:
4928
Disease MeSH ID:
-
Disease NCIt ID:
C35417
Disease ICD11 ID:
1253728223; 387909164
Disease OMIM ID:
-
Species: Human
Species details: Homo sapiens
Tissue specimen:

ICC tumor tissues; adjacent normal tissues; xenograft tumor tissues

Cell lines:

RBE; HCCC-9810; QBC-939; HUCCT1; HIBEC

In vivo animal model:

cell line-derived xenograft

circRNA-disease information
Expression pattern:
UP
Associated gene: PDK1, pyruvate dehydrogenase kinase 1
Associated microRNA: miR-152-3p
Biological function: Facilitates ICC cell proliferation, invasion, migration, glycolysis and tumor growth, and inhibits apoptosis.
Molecular mechanism: circ_0000284 acts as a ceRNA sponge for miR-152-3p to upregulate PDK1 expression, promoting ICC growth, metastasis and glycolysis.
Biological pathway or process:

ceRNA regulation (promotes); proliferation (promotes); apoptosis (inhibits); migration (promotes); invasion (promotes); metastasis (promotes); glycolysis (promotes)

Detected method:
Q
Validation methods:

RNase R Treatment; RT-qPCR; Clinical Sample Validation; Nuclear-Cytoplasmic Fractionation; Transfection; CCK8; EdU Staining; Annexin V/PI Flow Cytometry; Transwell Assay; Wound Healing Assay; Western Blot; Luciferase Reporter Assay; Bioinformatics Analysis; IHC (Immunohistochemistry); In Vivo Animal Model; H&E Staining; Survival Analysis; Cohort Study

Clinical significance:

High circ_0000284 expression was associated with lower overall survival rate and lymph node metastasis in ICC patients.

Description:

circ_0000284 is up-regulated in ICC tissues and cells and is associated with lymph node metastasis and poorer overall survival. Functionally, it promotes ICC proliferation, invasion, migration, glycolysis and xenograft tumor growth while suppressing apoptosis. Mechanistically, circ_0000284 acts as a cytoplasmic ceRNA sponge for miR-152-3p, thereby increasing PDK1 expression and driving ICC malignant progression.

Confidence score:

0.8157

Other information
Title:

Circ_0000284 facilitates the growth, metastasis and glycolysis of intrahepatic cholangiocarcinoma through miR-152-3p-mediated PDK1 expression.

Journal: Histology and histopathology
Published: 2023
PubMed ID: 36331285
Study type:

combined biological and clinical study

Data availability: The analyzed data sets generated during the present study are available from the corresponding author on reasonable request.
Code availability: -