circRNA basic information
circBase ID: hsa_circ_0017114
Name: hsa_circ_GPR137B
Synonym: circGPR137B / circ_0017114
Host Gene: GPR137B
Genomic location(hg19): chr1:236332005-236372209:+
Genomic location(hg38): chr1:236168705-236208909:+
Subcellular localization: cytoplasm
 
 
 
 
 
 
 
Disease basic information
MONDO ID:
0007256
MONDO name: hepatocellular carcinoma
Disease details: hepatocellular carcinoma / HCC
Disease DO ID:
684, 686
Disease MeSH ID:
D006528
Disease NCIt ID:
C3099
Disease ICD11 ID:
1294035808
Disease OMIM ID:
114550
Species: Human
Species details: Homo sapiens
Tissue specimen:

HCC tissues; adjacent normal tissues; frozen HCC tissue samples; tissue microarray

Cell lines:

HepG2; Hep3B; SK-hep-1; LO2; Huh6; Huh7

In vivo animal model:

cell line-derived xenograft

circRNA-disease information
Expression pattern:
DN
Associated gene: FTO, Ago2
Associated microRNA: miR-4739
Biological function: inhibits proliferation, colony formation, invasion, tumor growth and lung metastasis
Molecular mechanism: circGPR137B sponges miR-4739 to upregulate FTO; FTO binds circGPR137B and demethylates m6A to promote circGPR137B expression, forming a positive feedback loop
Biological pathway or process:

proliferation (inhibits); invasion (inhibits); metastasis (inhibits); ceRNA regulation (other); m6A modification (other)

Detected method:
Q
H
M
Validation methods:

Microarray; RT-qPCR; FISH / smFISH; Nuclear-Cytoplasmic Fractionation; RNase R Treatment; Actinomycin D / DRB Stability Assay; Luciferase Reporter Assay; RIP (RNA Immunoprecipitation); MeRIP / MeRIP-seq; Transfection; MTT; Colony Formation Assay; Transwell Assay; Western Blot; In Vivo Animal Model; H&E Staining; IHC (Immunohistochemistry); Clinical Sample Validation; Cohort Study; Survival Analysis; Bioinformatics Analysis

Clinical significance:

downregulation of circGPR137B was associated with poor prognosis in patients with HCC

Description:

circGPR137B is down-regulated in HCC and functions as a tumor suppressor. It sponges miR-4739 to relieve repression of FTO, while FTO demethylates circGPR137B (m6A) and enhances circGPR137B expression, forming a positive feedback loop that inhibits proliferation, invasion, and metastasis.

Confidence score:

0.8846

Other information
Title:

CircGPR137B/miR-4739/FTO feedback loop suppresses tumorigenesis and metastasis of hepatocellular carcinoma.

Journal: Molecular cancer
Published: 2022
PubMed ID: 35858900
Study type:

combined biological and clinical study

Data availability: -
Code availability: -