circRNA basic information
circBase ID: -
Name: hsa_circ_KEAP1
Synonym: circKEAP1
Host Gene: KEAP1
Genomic location(hg19): -
Genomic location(hg38): -
Subcellular localization: cytoplasm
 
 
 
 
 
 
 
Disease basic information
MONDO ID:
0005061
MONDO name: lung adenocarcinoma
Disease details: lung adenocarcinoma
Disease DO ID:
3910
Disease MeSH ID:
C538231
Disease NCIt ID:
C3512
Disease ICD11 ID:
-
Disease OMIM ID:
-
Species: Human
Species details: Homo sapiens
Tissue specimen:

LUAD cancer tissues; adjacent normal tissues

Cell lines:

BEAS-2B; A549; PC9; H1975

In vivo animal model:

cell line-derived xenograft

circRNA-disease information
Expression pattern:
DN
Associated gene: KEAP1, NRF2, HDAC4, AGO2
Associated microRNA: miR-141-3p
Biological function: Suppresses LUAD progression by inhibiting tumor growth, proliferation and migration.
Molecular mechanism: Acts as a ceRNA/miRNA sponge: circKEAP1 binds miR-141-3p to relieve repression on KEAP1, modulating the KEAP1/NRF2/HDAC4 signaling pathway.
Biological pathway or process:

proliferation (inhibits); migration (inhibits); KEAP1/NRF2/HDAC4 signal pathway (inhibits); ceRNA regulation (promotes)

Detected method:
Q
B
M
Validation methods:

Microarray; RT-qPCR; Back-Splice Junction PCR / divergent primers PCR; Sanger Sequencing; Northern Blot; Nuclear-Cytoplasmic Fractionation; Actinomycin D / DRB Stability Assay; Luciferase Reporter Assay; RNA Pull-Down; RIP (RNA Immunoprecipitation); Transfection; CCK8; MTT; EdU Staining; Transwell Assay; In Vivo Animal Model; H&E Staining; IHC (Immunohistochemistry); Western Blot; Clinical Sample Validation; Cohort Study; Survival Analysis; Bioinformatics Analysis

Clinical significance:

Low circKEAP1 was associated with unfavorable prognosis and correlated with lymphatic metastasis and tumor stage.

Description:

circKEAP1 (hsa_circRNA_102442) is down-regulated in LUAD and functions as a tumor suppressor. It sponges miR-141-3p to de-repress KEAP1, thereby modulating the KEAP1/NRF2/HDAC4 signaling cascade and inhibiting LUAD cell proliferation/migration and xenograft growth. Low circKEAP1 expression is associated with unfavorable prognosis in LUAD patients.

Confidence score:

0.8942

Other information
Title:

CircKEAP1 Suppresses the Progression of Lung Adenocarcinoma via the miR-141-3p/KEAP1/NRF2 Axis.

Journal: Frontiers in oncology
Published: 2021
PubMed ID: 34136401
Study type:

combined biological and clinical study

Data availability: GSE112214; GSE101586; https://www.frontiersin.org/articles/10.3389/fonc.2021.672586/full#supplementary-material
Code availability: -