circRNA basic information
circBase ID: hsa_circ_0002483
Name: hsa_circ_PTK2
Synonym: circPTK2
Host Gene: PTK2
Genomic location(hg19): chr8:141874410-141900868:-
Genomic location(hg38): chr8:140864311-140890769:-
Subcellular localization: not tested
 
 
 
 
 
 
 
Disease basic information
MONDO ID:
0018874
MONDO name: acute myeloid leukemia
Disease details: acute myeloid leukemia
Disease DO ID:
9119
Disease MeSH ID:
D015470
Disease NCIt ID:
C3171
Disease ICD11 ID:
-
Disease OMIM ID:
601626
Species: Human
Species details: Homo sapiens
Tissue specimen:

peripheral blood samples

Cell lines:

HS-5; HL-60; KG-1

In vivo animal model:

-

circRNA-disease information
Expression pattern:
UP
Associated gene: ALG3, Ago2
Associated microRNA: miR-582-3p
Biological function: CircPTK2 promotes AML cell viability, proliferation, cell cycle process and glycolysis, and inhibits apoptosis; circPTK2 knockdown suppresses malignant biological behaviors of AML cells.
Molecular mechanism: CircPTK2 acts as a ceRNA/sponge for miR-582-3p, thereby positively regulating ALG3 expression in AML cells.
Biological pathway or process:

proliferation (promotes); cell cycle (promotes); glycolysis (promotes); apoptosis (inhibits); ceRNA regulation (other)

Detected method:
Q
Validation methods:

RT-qPCR; Clinical Sample Validation; Transfection; MTT; EdU Staining; Annexin V/PI Flow Cytometry; Cell Cycle Assay; Western Blot; Luciferase Reporter Assay; RIP (RNA Immunoprecipitation); Bioinformatics Analysis

Clinical significance:

CircPTK2 is upregulated in AML peripheral blood samples and might provide a potential target for AML therapy.

Description:

CircPTK2 is upregulated in AML peripheral blood samples and AML cell lines. Functionally, circPTK2 promotes AML cell viability, proliferation, cell cycle progression and glycolysis while suppressing apoptosis. Mechanistically, it acts as a sponge for miR-582-3p to positively regulate ALG3 expression, forming a circPTK2/miR-582-3p/ALG3 axis that contributes to AML malignant behaviors.

Confidence score:

0.7045

Other information
Title:

CircPTK2 promotes cell viability, cell cycle process, and glycolysis and inhibits cell apoptosis in acute myeloid leukemia by regulating miR-582-3p/ALG3 axis.

Journal: Expert review of hematology
Published: 2022
PubMed ID: 35980117
Study type:

combined biological and clinical study

Data availability: The analyzed data sets generated during the present study are available from the corresponding author on reasonable request.
Code availability: -