circRNA basic information
circBase ID: hsa_circ_0001666
Name: -
Synonym: circ_0001666
Host Gene: -
Genomic location(hg19): chr6:170626457-170639638:+
Genomic location(hg38): chr6:170317369-170330550:+
Subcellular localization: cytoplasm
 
 
 
 
 
 
 
Disease basic information
MONDO ID:
0007254
MONDO name: breast cancer
Disease details: breast cancer
Disease DO ID:
1612
Disease MeSH ID:
-
Disease NCIt ID:
C9335
Disease ICD11 ID:
1047754165
Disease OMIM ID:
-
Species: Human
Species details: Homo sapiens
Tissue specimen:

BC tumor tissues; paracarcinoma tissues; non-tumor tissues

Cell lines:

MCF-10A; MDA-MB-231; MDA-MB-453; BT20; MCF-7; SK-BR-3

In vivo animal model:

cell line-derived xenograft

circRNA-disease information
Expression pattern:
DN
Associated gene: WNK2
Associated microRNA: miR-620
Biological function: Circ_0001666 acts as a tumor suppressor in breast cancer, inhibiting cell proliferation, migration, invasion, metastasis-related phenotypes and tumor growth, while promoting apoptosis and inducing G0/G1 cell-cycle arrest.
Molecular mechanism: Circ_0001666 functions through a ceRNA mechanism by sponging miR-620, thereby positively regulating WNK2 expression and inhibiting breast cancer progression.
Biological pathway or process:

proliferation (inhibits); migration (inhibits); invasion (inhibits); metastasis (inhibits); apoptosis (promotes); cell cycle (inhibits); ceRNA regulation (other)

Detected method:
Q
M
Validation methods:

RT-qPCR; RNase R Treatment; Nuclear-Cytoplasmic Fractionation; Clinical Sample Validation; Bioinformatics Analysis; Transfection; CCK8; Annexin V/PI Flow Cytometry; Cell Cycle Assay; Transwell Assay; Western Blot; Luciferase Reporter Assay; RIP (RNA Immunoprecipitation); In Vivo Animal Model

Clinical significance:

circ_0001666 expression was related to tumor size, TNM stage and lymph node metastases in breast cancer patients, and the authors proposed it as a new target for targeted therapy of breast cancer.

Description:

This study identified circ_0001666 as a downregulated circRNA in breast cancer tissues and cell lines. Functional assays showed that circ_0001666 suppresses breast cancer progression by inhibiting proliferation, migration, invasion, metastasis-related phenotypes and tumor growth, while promoting apoptosis. Mechanistically, circ_0001666 acts as a miR-620 sponge to upregulate WNK2 in a circ_0001666/miR-620/WNK2 ceRNA axis.

Confidence score:

0.7799

Other information
Title:

Circ_0001666 affects miR-620/WNK2 axis to inhibit breast cancer progression.

Journal: Genes & genomics
Published: 2021
PubMed ID: 34061329
Study type:

combined biological and clinical study

Data availability: GSE112214; GSE101124; supplementary material available at https://doi.org/10.1007/s13258-021-01114-y; analyzed data sets generated during the present study are available from the corresponding author on reasonable request
Code availability: -