circRNA basic information
circBase ID: hsa_circ_0000419
Name: hsa_circ_RAB3IP
Synonym: circRAB3IP
Host Gene: RAB3IP
Genomic location(hg19): chr12:70193988-70195501:+
Genomic location(hg38): chr12:69800208-69801721:+
Subcellular localization: cytoplasm
 
 
 
 
 
 
 
Disease basic information
MONDO ID:
0008315
MONDO name: prostate cancer
Disease details: prostate cancer
Disease DO ID:
10283
Disease MeSH ID:
D011471
Disease NCIt ID:
C7378
Disease ICD11 ID:
-
Disease OMIM ID:
-
Species: Human
Species details: Homo sapiens
Tissue specimen:

prostate tissue

Cell lines:

22Rv1; C4-2; C4-2-EnzR; LNCaP; LNCaP-EnzR; 293T

In vivo animal model:

cell line-derived xenograft

circRNA-disease information
Expression pattern:
UP
Associated gene: SGK1, eIF4A3, LEF1, AGO2
Associated microRNA: miR-133a-3p, miR-133b
Biological function: promotes enzalutamide resistance and decreases enzalutamide sensitivity; promotes cell proliferation/viability under enzalutamide treatment
Molecular mechanism: Acts as a ceRNA/miRNA sponge for miR-133a-3p and miR-133b to upregulate SGK1; biogenesis promoted by eIF4A3 (binding flanking pre-mRNA) and LEF1 (transcriptionally regulates RAB3IP promoter).
Biological pathway or process:

chemoresistance (promotes); proliferation (promotes); ceRNA regulation (promotes)

Detected method:
Q
S
M
Validation methods:

Microarray; RNA-seq; RT-qPCR; divergent primers PCR; RNase R Treatment; Actinomycin D / DRB Stability Assay; Nuclear-Cytoplasmic Fractionation; FISH / smFISH; RIP (RNA Immunoprecipitation); RNA Pull-Down; Luciferase Reporter Assay; Transfection; MTT; CCK8; Western Blot; ChIP / ChIP-seq; In Vivo Animal Model; Bioinformatics Analysis; Clinical Sample Validation

Clinical significance:

circRAB3IP expression was significantly upregulated in EnzR PCa tissues compared with EnzS PCa tissues; higher in high grade PCa than low grade PCa or BPH

Description:

circRAB3IP (hsa_circ_0000419), derived from RAB3IP, is upregulated in enzalutamide-resistant prostate cancer cells and tissues and promotes enzalutamide resistance. It mainly localizes to the cytoplasm and acts as a ceRNA by sponging miR-133a-3p/miR-133b to increase SGK1 expression; its expression/biogenesis is promoted by eIF4A3 and LEF1.

Confidence score:

0.8575

Other information
Title:

The circRAB3IP Mediated by eIF4A3 and LEF1 Contributes to Enzalutamide Resistance in Prostate Cancer by Targeting miR-133a-3p/miR-133b/SGK1 Pathway.

Journal: Frontiers in oncology
Published: 2021
PubMed ID: 34868959
Study type:

combined biological and clinical study

Data availability: GSE118959; GSE104935; Supplementary Material: https://www.frontiersin.org/articles/10.3389/fonc.2021.752573/full#supplementary-material
Code availability: -