circRNA basic information
circBase ID: hsa_circ_0004650
Name: -
Synonym: -
Host Gene: -
Genomic location(hg19): chr12:47497895-47501947:+
Genomic location(hg38): chr12:47104112-47108164:+
Subcellular localization: not tested
 
 
 
 
 
 
 
Disease basic information
MONDO ID:
0001056
MONDO name: gastric cancer
Disease details: gastric cancer
Disease DO ID:
10534
Disease MeSH ID:
-
Disease NCIt ID:
C9331
Disease ICD11 ID:
1397617262
Disease OMIM ID:
613659
Species: Human
Species details: Homo sapiens
Tissue specimen:

-

Cell lines:

SGC-7901; BGC-823; SGC-7901-5-Fu; BGC-823-5-Fu; HEK-293T

In vivo animal model:

-

circRNA-disease information
Expression pattern:
UP
Associated gene: -
Associated microRNA: miR-145-5p
Biological function: Promotes 5-Fu resistance in gastric cancer cells; silencing hsa_circ_0004650 decreases cell survival/proliferation activity and promotes apoptosis under 5-Fu treatment.
Molecular mechanism: hsa_circ_0004650 functions as a ceRNA/miRNA sponge that targets and negatively regulates miR-145-5p, thereby inhibiting apoptosis and facilitating 5-Fu resistance in gastric cancer cells.
Biological pathway or process:

drug resistance (promotes); chemoresistance (promotes); proliferation (promotes); apoptosis (inhibits); ceRNA regulation (other)

Detected method:
Q
S
Validation methods:

RT-qPCR; RNA-seq; Bioinformatics Analysis; Luciferase Reporter Assay; Transfection; CCK8; Annexin V/PI Flow Cytometry

Clinical significance:

Potential therapeutic target for overcoming 5-Fu resistance in gastric cancer.

Description:

hsa_circ_0004650 is up-regulated in 5-Fu-resistant gastric cancer cell lines. It promotes 5-Fu resistance by sponging and negatively regulating miR-145-5p, thereby enhancing cell survival/proliferation and inhibiting apoptosis under 5-Fu treatment. The study proposes hsa_circ_0004650 as a potential therapeutic target for overcoming 5-Fu resistance in gastric cancer.

Confidence score:

0.5804

Other information
Title:

Circular RNA hsa_circ_0004650 Enhances 5-Fluorouracil Resistance in Gastric Cancer via Sponging miR-145-5p.

Journal: Anticancer research
Published: 2024
PubMed ID: 39740828
Study type:

biological research

Data availability: Dryad: https://Datadryad.org/stash/dataset/doi:10.5061/dryad.v15dv41wv
Code availability: -