circRNA basic information
circBase ID: hsa_circ_0058124
Name: hsa_circ_FN1
Synonym: circFN1
Host Gene: FN1
Genomic location(hg19): chr2:216270960-216274462:-
Genomic location(hg38): chr2:215406237-215409739:-
Subcellular localization: cytoplasm
 
 
 
 
 
 
 
Disease basic information
MONDO ID:
0007256
MONDO name: hepatocellular carcinoma
Disease details: hepatocellular carcinoma
Disease DO ID:
684, 686
Disease MeSH ID:
D006528
Disease NCIt ID:
C3099
Disease ICD11 ID:
1294035808
Disease OMIM ID:
114550
Species: Human
Species details: Homo sapiens
Tissue specimen:

HCC tissues; paired adjacent normal tissues (ANTs); xenograft tumor tissue

Cell lines:

HepG2; Huh-7; LO2; SR-HepG2; SR-Huh7

In vivo animal model:

cell line-derived xenograft

circRNA-disease information
Expression pattern:
UP
Associated gene: E2F1, AGO2
Associated microRNA: miR-1205
Biological function: promotes sorafenib resistance, promotes proliferation, inhibits apoptosis in HCC cells
Molecular mechanism: Acts as a ceRNA/miRNA sponge for miR-1205 to upregulate E2F1 expression, contributing to sorafenib resistance
Biological pathway or process:

chemoresistance (promotes); proliferation (promotes); apoptosis (inhibits); ceRNA regulation (promotes); PI3K/AKT (promotes)

Detected method:
Q
M
Validation methods:

Microarray; RT-qPCR; RNase R Treatment; Actinomycin D / DRB Stability Assay; Nuclear-Cytoplasmic Fractionation; Transfection; CCK8; Annexin V/PI Flow Cytometry; In Vivo Animal Model; IHC (Immunohistochemistry); RIP (RNA Immunoprecipitation); RNA Pull-Down; Luciferase Reporter Assay; Western Blot; Clinical Sample Validation; Cohort Study; Survival Analysis; ROC Analysis; Bioinformatics Analysis

Clinical significance:

High circFN1 expression was associated with tumor size, TNM stage, vascular invasion, and shorter overall survival; ROC AUC 0.878 for distinguishing HCC tissues from ANTs

Description:

circFN1 (hsa_circ_0058124) is upregulated in HCC tissues and sorafenib-resistant HCC cells, and its high expression predicts poorer overall survival. Functionally, circFN1 promotes proliferation and sorafenib resistance while inhibiting sorafenib-induced apoptosis, at least partly by sponging miR-1205 to increase E2F1 expression.

Confidence score:

0.8837

Other information
Title:

circFN1 Mediates Sorafenib Resistance of Hepatocellular Carcinoma Cells by Sponging miR-1205 and Regulating E2F1 Expression.

Journal: Molecular therapy. Nucleic acids
Published: 2020
PubMed ID: 33230446
Study type:

combined biological and clinical study

Data availability: Supplemental Information can be found online at https://doi.org/10.1016/j.omtn.2020.08.039
Code availability: -