circRNA basic information
circBase ID: hsa_circ_0001667
Name: hsa_circ_HEATR2
Synonym: circ_0001667
Host Gene: -
Genomic location(hg19): chr7:810107-814799:+
Genomic location(hg38): chr7:770470-775162:+
Subcellular localization: cytoplasm
 
 
 
 
 
 
 
Disease basic information
MONDO ID:
0007254
MONDO name: breast cancer
Disease details: breast cancer
Disease DO ID:
1612
Disease MeSH ID:
-
Disease NCIt ID:
C9335
Disease ICD11 ID:
1047754165
Disease OMIM ID:
-
Species: Human
Species details: Homo sapiens
Tissue specimen:

breast cancer tissues; normal tissues; tumor tissues

Cell lines:

MCF-7; MDA-MB-231; MCF-7/ADM; MDA-MB-231/ADM

In vivo animal model:

cell line-derived xenograft

circRNA-disease information
Expression pattern:
UP
Associated gene: NCOA3
Associated microRNA: miR-4458
Biological function: Circ_0001667 promotes ADM-resistant breast cancer cell proliferation, migration, invasion, tumor growth and ADM resistance, and inhibits ADM-induced apoptosis; circ_0001667 knockdown suppresses these malignant behaviors and attenuates ADM resistance.
Molecular mechanism: Circ_0001667 acts as a ceRNA/miRNA sponge for miR-4458, thereby relieving miR-4458-mediated repression of NCOA3 and promoting ADM resistance and malignant progression.
Biological pathway or process:

proliferation (promotes); migration (promotes); invasion (promotes); apoptosis (inhibits); drug resistance (promotes); chemoresistance (promotes); ceRNA regulation (other); other pathway/process (promotes)

Detected method:
Q
Validation methods:

RNase R Treatment; RT-qPCR; Clinical Sample Validation; Nuclear-Cytoplasmic Fractionation; Transfection; MTT; Colony Formation Assay; Transwell Assay; Western Blot; Annexin V/PI Flow Cytometry; Bioinformatics Analysis; RNA Pull-Down; Luciferase Reporter Assay; RIP (RNA Immunoprecipitation); In Vivo Animal Model; IHC (Immunohistochemistry)

Clinical significance:

-

Description:

Circ_0001667 is up-regulated in ADM-resistant breast cancer tissues and cells. Its knockdown suppresses proliferation, migration, invasion, tumor growth and ADM resistance while promoting ADM-induced apoptosis. Mechanistically, circ_0001667 functions through the circ_0001667/miR-4458/NCOA3 axis, acting as a miR-4458 sponge to maintain NCOA3 expression and promote chemoresistant malignant progression.

Confidence score:

0.8324

Other information
Title:

Circ_0001667 knockdown blocks cancer progression and attenuates adriamycin resistance by depleting NCOA3 via releasing miR-4458 in breast cancer.

Journal: Drug development research
Published: 2022
PubMed ID: 34227151
Study type:

combined biological and clinical study

Data availability: -
Code availability: -