circRNA basic information
circBase ID: -
Name: hsa_circ_XIAP
Synonym: circ-XIAP
Host Gene: XIAP
Genomic location(hg19): -
Genomic location(hg38): -
Subcellular localization: cytoplasm; exosome
 
 
 
 
 
 
 
Disease basic information
MONDO ID:
0008315
MONDO name: prostate cancer
Disease details: prostate cancer
Disease DO ID:
10283
Disease MeSH ID:
D011471
Disease NCIt ID:
C7378
Disease ICD11 ID:
-
Disease OMIM ID:
-
Species: Human
Species details: Homo sapiens
Tissue specimen:

PCa tissue specimens; tumor tissues; adjacent normal tissues

Cell lines:

22Rv1; VCaP; DU145; PC3; RWPE-1; DU145/DTX; PC3/DTX

In vivo animal model:

cell line-derived xenograft

circRNA-disease information
Expression pattern:
UP
Associated gene: TPD52
Associated microRNA: miR-1182
Biological function: promotes docetaxel resistance, proliferation, migration and invasion, and inhibits apoptosis and G0/G1 cell cycle arrest in DTX-resistant PCa cells; promotes tumor growth and reduces DTX sensitivity in vivo
Molecular mechanism: Exosomal circ-XIAP acts as a miRNA sponge for miR-1182, thereby upregulating TPD52 and promoting docetaxel resistance (ceRNA mechanism).
Biological pathway or process:

chemoresistance (promotes); proliferation (promotes); migration (promotes); invasion (promotes); apoptosis (inhibits); cell cycle (other); ceRNA regulation (promotes)

Detected method:
Q
Validation methods:

RT-qPCR; RNase R Treatment; Nuclear-Cytoplasmic Fractionation; Western Blot; Luciferase Reporter Assay; Transfection; CCK8; Colony Formation Assay; Cell Cycle Assay; Annexin V/PI Flow Cytometry; Transwell Assay; IHC (Immunohistochemistry); In Vivo Animal Model; Bioinformatics Analysis

Clinical significance:

-

Description:

circ-XIAP is upregulated in docetaxel-resistant prostate cancer tissues/cells and enriched in exosomes. It promotes DTX resistance by acting as a sponge for miR-1182, thereby increasing TPD52 expression, enhancing malignant phenotypes and reducing chemosensitivity in vitro and in a xenograft model.

Confidence score:

0.7421

Other information
Title:

Exosomal Circ-XIAP Promotes Docetaxel Resistance in Prostate Cancer by Regulating miR-1182/TPD52 Axis.

Journal: Drug design, development and therapy
Published: 2021
PubMed ID: 33976535
Study type:

combined biological and clinical study

Data availability: -
Code availability: -