circRNA basic information
circBase ID: -
Name: hsa_circ_PITX1
Synonym: -
Host Gene: PITX1
Genomic location(hg19): -
Genomic location(hg38): -
Subcellular localization: not tested
 
 
 
 
 
 
 
Disease basic information
MONDO ID:
0021042
MONDO name: glioma
Disease details: glioma
Disease DO ID:
-
Disease MeSH ID:
D005910
Disease NCIt ID:
C3059
Disease ICD11 ID:
-
Disease OMIM ID:
-
Species: Human
Species details: Homo sapiens
Tissue specimen:

glioma tissues; normal brain tissues

Cell lines:

U251; LN229; NHA

In vivo animal model:

cell line-derived xenograft

circRNA-disease information
Expression pattern:
UP
Associated gene: NEK2
Associated microRNA: miR-329-3p
Biological function: Promotes glycolysis and radioresistance; promotes cell viability and clonogenic survival; promotes tumor growth in vivo; circPITX1 knockdown enhances radiosensitivity.
Molecular mechanism: Acts as a ceRNA to sponge miR-329-3p, thereby relieving repression of NEK2 and promoting glycolysis-associated factors (HIF-1alpha, HK2, LDH-A) and radioresistance.
Biological pathway or process:

glycolysis (promotes); radioresistance (promotes); proliferation (promotes)

Detected method:
Q
Validation methods:

RT-qPCR; RNase R Treatment; Western Blot; Luciferase Reporter Assay; Transfection; MTT; Colony Formation Assay; In Vivo Animal Model; Bioinformatics Analysis; Clinical Sample Validation

Clinical significance:

-

Description:

circPITX1 is up-regulated in glioma tissues/cells and promotes glycolysis and radioresistance. Mechanistically, circPITX1 sponges miR-329-3p to increase NEK2 expression, enhancing glycolysis-associated protein expression and clonogenic survival; circPITX1 knockdown inhibits tumor growth in xenografts and increases radiosensitivity.

Confidence score:

0.7164

Other information
Title:

Circular RNA circPITX1 knockdown inhibits glycolysis to enhance radiosensitivity of glioma cells by miR-329-3p/NEK2 axis.

Journal: Cancer cell international
Published: 2020
PubMed ID: 32190004
Study type:

combined biological and clinical study

Data availability: All data generated or analyzed during this study are included in this published article.
Code availability: -