circRNA basic information
circBase ID: hsa_circ_0097922
Name: hsa_circ_PGAM5
Synonym: Circ_0097922
Host Gene: PGAM5
Genomic location(hg19): -
Genomic location(hg38): -
Subcellular localization: cytoplasm
 
 
 
 
 
 
 
Disease basic information
MONDO ID:
0007254
MONDO name: breast cancer
Disease details: breast cancer
Disease DO ID:
1612
Disease MeSH ID:
-
Disease NCIt ID:
C9335
Disease ICD11 ID:
1047754165
Disease OMIM ID:
-
Species: Human
Species details: Homo sapiens
Tissue specimen:

BC tissues; normal tissues; tumour tissues; xenograft tumour tissues

Cell lines:

MCF7; T47D; MCF7/TR; T47D/TR; HEK293T; MCT-10A

In vivo animal model:

cell line-derived xenograft

circRNA-disease information
Expression pattern:
UP
Associated gene: ACTN4, AGO2, PGAM5
Associated microRNA: miR-876-3p
Biological function: Promotes tamoxifen resistance, tumour growth, cell survival, proliferation, migration and invasion, and inhibits apoptosis in breast cancer cells.
Molecular mechanism: ceRNA mechanism: hsa_circ_0097922 acts as a miR-876-3p sponge to regulate ACTN4 expression, thereby promoting malignant behaviour and tamoxifen resistance.
Biological pathway or process:

ceRNA regulation (promotes); drug resistance (promotes); proliferation (promotes); apoptosis (inhibits); migration (promotes); invasion (promotes)

Detected method:
Q
S
Validation methods:

RNase R Treatment; Actinomycin D / DRB Stability Assay; RT-qPCR; Clinical Sample Validation; Nuclear-Cytoplasmic Fractionation; RIP (RNA Immunoprecipitation); RNA Pull-Down; Luciferase Reporter Assay; Transfection; CCK8; EdU Staining; Colony Formation Assay; Annexin V/PI Flow Cytometry; Transwell Assay; Wound Healing Assay; Western Blot; In Vivo Animal Model; IHC (Immunohistochemistry); Bioinformatics Analysis

Clinical significance:

hsa_circ_0097922 expression was associated with TNM stage and may be a promising therapeutic target/preclinical basis for drug-resistant breast cancer patients.

Description:

hsa_circ_0097922 is up-regulated in breast cancer tissues and tamoxifen-resistant breast cancer cells. It promotes malignant phenotypes and tamoxifen resistance by sponging miR-876-3p and increasing ACTN4 expression, while its knockdown sensitizes resistant cells and xenograft tumors to tamoxifen.

Confidence score:

0.8572

Other information
Title:

Hsa_circ_0097922 promotes tamoxifen resistance and cell malignant behaviour of breast cancer cells by regulating ACTN4 expression via miR-876-3p.

Journal: Clinical and experimental pharmacology & physiology
Published: 2022
PubMed ID: 35856314
Study type:

combined biological and clinical study

Data availability: The datasets generated during and analysed during the current study are available from the corresponding author on reasonable request.
Code availability: -