circRNA basic information
circBase ID: -
Name: hsa_circ_HIPK2
Synonym: -
Host Gene: HIPK2
Genomic location(hg19): -
Genomic location(hg38): -
Subcellular localization: cytoplasm
 
 
 
 
 
 
 
Disease basic information
MONDO ID:
0005575
MONDO name: colorectal cancer
Disease details: colorectal cancer / CRC
Disease DO ID:
5672, 9256
Disease MeSH ID:
-
Disease NCIt ID:
C4978
Disease ICD11 ID:
-
Disease OMIM ID:
114500
Species: Human
Species details: Homo sapiens
Tissue specimen:

cancer tissue; paracancerous tissue; serum samples

Cell lines:

NCM460; HCT-116; HT-29; COLO 25; SW480; HEK293T

In vivo animal model:

-

circRNA-disease information
Expression pattern:
UP
Associated gene: HSP90
Associated microRNA: miR-485-5p
Biological function: circHIPK2 promotes CRC progression, cell proliferation, EdU-positive cell rate, and migration, and its downregulation inhibits these malignant phenotypes.
Molecular mechanism: circHIPK2 is mainly cytoplasmic and regulates the miR-485-5p/HSP90 axis; circHIPK2 suppresses miR-485-5p, induces HSP90 expression, and promotes CRC tumor growth and progression via HSP90 ubiquitination.
Biological pathway or process:

proliferation (promotes); migration (promotes); ubiquitination (promotes); ceRNA regulation (other)

Detected method:
Q
S
M
Validation methods:

RT-qPCR; RNA-seq; Microarray; FISH / smFISH; Nuclear-Cytoplasmic Fractionation; Clinical Sample Validation; Luciferase Reporter Assay; Transfection; CCK8; EdU Staining; Western Blot; IF (Immunofluorescence); Survival Analysis

Clinical significance:

circHIPK2 is upregulated in CRC patients, high circHIPK2 expression is associated with lower overall survival and disease-free survival, and circHIPK2 is considered a promising biomarker for CRC diagnosis and prognosis and a potential therapeutic target.

Description:

circHIPK2 is upregulated in CRC tissues and cell lines and high expression is associated with poorer overall and disease-free survival. Functionally, circHIPK2 promotes CRC cell proliferation and migration, likely through a cytoplasmic circHIPK2/miR-485-5p/HSP90 regulatory mechanism involving HSP90 ubiquitination. The study proposes circHIPK2 as a potential diagnostic/prognostic biomarker and therapeutic target for CRC.

Confidence score:

0.7357

Other information
Title:

circHIPK2 Has a Potentially Important Clinical Significance in Colorectal Cancer Progression via HSP90 Ubiquitination by miR485-5p.

Journal: Critical reviews in eukaryotic gene expression
Published: 2022
PubMed ID: 36017914
Study type:

combined biological and clinical study

Data availability: -
Code availability: -