circRNA basic information
circBase ID: -
Name: hsa_circ_AKT3
Synonym: Circular RNA AKT3 / CircAKT3
Host Gene: AKT3
Genomic location(hg19): -
Genomic location(hg38): -
Subcellular localization: not tested
 
 
 
 
 
 
 
Disease basic information
MONDO ID:
0008903
MONDO name: lung cancer
Disease details: lung cancer
Disease DO ID:
1324
Disease MeSH ID:
-
Disease NCIt ID:
C7377
Disease ICD11 ID:
-
Disease OMIM ID:
211980
Species: Human
Species details: Homo sapiens
Tissue specimen:

lung cancer tissues; normal adjacent tissue

Cell lines:

A549; H1299; BEAS-2B

In vivo animal model:

cell line-derived xenograft

circRNA-disease information
Expression pattern:
UP
Associated gene: STAT3, HIF-1a
Associated microRNA: miR-516b-5p
Biological function: circAKT3 promotes cisplatin resistance, HIF-1a-dependent glycolysis and tumor growth in lung cancer; knockdown of circAKT3 increases cisplatin sensitivity, represses glycolysis and suppresses xenograft tumor growth.
Molecular mechanism: circAKT3 acts through the miR-516b-5p/STAT3 axis to regulate HIF-1a-dependent glycolysis and cisplatin sensitivity.
Biological pathway or process:

glycolysis (promotes); chemoresistance (promotes); proliferation (promotes); ceRNA regulation (other)

Detected method:
Q
Validation methods:

RT-qPCR; Clinical Sample Validation; Transfection; MTT; Luciferase Reporter Assay; Western Blot; In Vivo Animal Model; Bioinformatics Analysis

Clinical significance:

These findings provided new insights and ideas for clinical prediction and treatment of lung cancer.

Description:

circAKT3 is up-regulated in lung cancer tissues and cell lines. It promotes cisplatin resistance and glycolysis, at least partly through regulation of the miR-516b-5p/STAT3 axis and HIF-1a-dependent glycolysis; circAKT3 knockdown increases cisplatin sensitivity and suppresses tumor growth in vivo.

Confidence score:

0.6479

Other information
Title:

CircAKT3 inhibits glycolysis balance in lung cancer cells by regulating miR-516b-5p/STAT3 to inhibit cisplatin sensitivity.

Journal: Biotechnology letters
Published: 2020
PubMed ID: 32170433
Study type:

combined biological and clinical study

Data availability: -
Code availability: -