circRNA basic information
circBase ID: hsa_circ_0084171
Name: hsa_circ_FNTA
Synonym: circFNTA / circ_0084171
Host Gene: FNTA
Genomic location(hg19): chr8:42914234-42932507:+
Genomic location(hg38): chr8:43059091-43077364:+
Subcellular localization: cytoplasm
 
 
 
 
 
 
 
Disease basic information
MONDO ID:
0004986
MONDO name: urinary bladder carcinoma
Disease details: bladder cancer / BCa
Disease DO ID:
4007
Disease MeSH ID:
-
Disease NCIt ID:
C4912
Disease ICD11 ID:
-
Disease OMIM ID:
-
Species: Human
Species details: Homo sapiens
Tissue specimen:

BCa tissues; adjacent para-tumor tissues; fresh BCa tissues; para-tumor tissues; mouse tumor tissues; lung metastatic foci

Cell lines:

SVHUC; T24; J82; 5637; UMUC3

In vivo animal model:

cell line-derived xenograft

circRNA-disease information
Expression pattern:
UP
Associated gene: AR, ADAR2, FNTA, KRAS, ERK1/2, MEK1/2
Associated microRNA: miR-370-3p, miR-328-5p, miR-920
Biological function: circFNTA promotes bladder cancer cell invasion, metastasis, and cisplatin chemo-resistance; depletion of circFNTA suppresses xenograft growth and lung metastasis and increases cisplatin chemo-sensitivity.
Molecular mechanism: AR represses ADAR2 to increase circFNTA; circFNTA sponges miR-370-3p to increase FNTA expression, thereby activating KRAS signaling and downstream ERK1/2 and MEK1/2 phosphorylation.
Biological pathway or process:

ERK (promotes); invasion (promotes); metastasis (promotes); drug resistance (promotes); chemoresistance (promotes); ceRNA regulation (promotes)

Detected method:
Q
H
Validation methods:

RT-qPCR; RNase R Treatment; FISH / smFISH; Clinical Sample Validation; RNA Pull-Down; Luciferase Reporter Assay; ChIP / ChIP-seq; Transfection; MTT; Transwell Assay; In Vivo Animal Model; H&E Staining; IHC (Immunohistochemistry); Western Blot; Bioinformatics Analysis

Clinical significance:

circFNTA is elevated in bladder cancer tissues and may be a therapeutic target to suppress BCa metastasis and increase cisplatin chemo-sensitivity.

Description:

circFNTA is up-regulated in bladder cancer tissues and cell lines. It promotes bladder cancer invasion, metastasis, and cisplatin chemo-resistance through an AR/ADAR2/circFNTA/miR-370-3p/FNTA/KRAS signaling axis, and circFNTA depletion suppresses tumor growth and lung metastasis in vivo.

Confidence score:

0.8322

Other information
Title:

Androgen receptor-regulated circFNTA activates KRAS signaling to promote bladder cancer invasion.

Journal: EMBO reports
Published: 2020
PubMed ID: 32052578
Study type:

combined biological and clinical study

Data availability: GSE92675
Code availability: -