circRNA basic information
circBase ID: hsa_circ_0014130
Name: hsa_circ_PIP5K1A
Synonym: Circular RNA PIP5K1A / circ-PIP5K1A
Host Gene: PIP5K1A
Genomic location(hg19): chr1:151206672-151212515:+
Genomic location(hg38): chr1:151234196-151240039:+
Subcellular localization: exosome
 
 
 
 
 
 
 
Disease basic information
MONDO ID:
0008170
MONDO name: ovarian cancer
Disease details: ovarian cancer / OC
Disease DO ID:
2394
Disease MeSH ID:
D010051
Disease NCIt ID:
C7431
Disease ICD11 ID:
685124533
Disease OMIM ID:
167000
Species: Human
Species details: Homo sapiens
Tissue specimen:

OC tissues; matched noncancer tissues; DDP-resistant OC tissues; DDP-sensitive OC tissues; tumor tissues

Cell lines:

OVCAR3; HEY; A2780; SKOV3; A2780/DDP; SKOV3/DDP; HCEREPiC

In vivo animal model:

cell line-derived xenograft

circRNA-disease information
Expression pattern:
UP
Associated gene: NFIB, PIP5K1A mRNA, Bcl-2, MMP9
Associated microRNA: miR-942-5p
Biological function: Promotes cisplatin resistance, proliferation, migration, invasion, cell cycle progression and tumor growth; inhibits apoptosis and cisplatin sensitivity in ovarian cancer.
Molecular mechanism: circ-PIP5K1A functions as a ceRNA sponge for miR-942-5p, thereby positively regulating NFIB expression; it is also packaged into exosomes and transferred between ovarian cancer cells.
Biological pathway or process:

ceRNA regulation (promotes); drug resistance (promotes); chemoresistance (promotes); proliferation (promotes); migration (promotes); invasion (promotes); apoptosis (inhibits); cell cycle (promotes); metastasis (promotes); other pathway/process (promotes)

Detected method:
Q
Validation methods:

RNase R Treatment; RT-qPCR; Clinical Sample Validation; Transfection; CCK8; Colony Formation Assay; Annexin V/PI Flow Cytometry; Cell Cycle Assay; EdU Staining; Transwell Assay; Western Blot; Luciferase Reporter Assay; In Vivo Animal Model; IHC (Immunohistochemistry); Bioinformatics Analysis

Clinical significance:

Provided a promising therapeutic target for preventing cisplatin resistance in ovarian cancer and a new insight into exosome-based therapeutics.

Description:

circ-PIP5K1A is up-regulated in ovarian cancer, especially in cisplatin-resistant tissues and cells. It promotes cisplatin resistance and malignant phenotypes by sponging miR-942-5p to increase NFIB expression, and its knockdown sensitizes ovarian cancer cells and xenograft tumors to cisplatin. The study also shows that circ-PIP5K1A can be packaged into exosomes and transferred from resistant cells to surrounding sensitive cells.

Confidence score:

0.7663

Other information
Title:

Knockdown of circ-PIP5K1A overcomes resistance to cisplatin in ovarian cancer by miR-942-5p/NFIB axis.

Journal: Anti-cancer drugs
Published: 2023
PubMed ID: 36730637
Study type:

combined biological and clinical study

Data availability: the data that support the findings of this study are available from the corresponding author upon reasonable request
Code availability: -