circRNA basic information
circBase ID: hsa_circ_0006608
Name: hsa_circ_PFKP
Synonym: -
Host Gene: PFKP
Genomic location(hg19): chr10:3160973-3162236:+
Genomic location(hg38): chr10:3118781-3120044:+
Subcellular localization: cytoplasm
 
 
 
 
 
 
 
Disease basic information
MONDO ID:
0005075
MONDO name: thyroid gland papillary carcinoma
Disease details: Papillary thyroid carcinoma
Disease DO ID:
3969
Disease MeSH ID:
-
Disease NCIt ID:
C4035
Disease ICD11 ID:
-
Disease OMIM ID:
-
Species: Human
Species details: Homo sapiens
Tissue specimen:

PTC tissues; matched normal tissues; thyroid cancer and adjacent paracarcinoma samples; adjacent normal tissues

Cell lines:

TPC-1; B-CPAP; HEK-293 T; Nthy-ori 3-1; HTori-3; KTC-1

In vivo animal model:

cell line-derived xenograft

circRNA-disease information
Expression pattern:
UP
Associated gene: SPRY4, p38 MAPK signaling pathway
Associated microRNA: miR-4516
Biological function: circPFKP inhibits PTC cell proliferation, colony formation, migration, and invasion under baseline conditions, but protects PTC cells from stress- or radiation-induced apoptosis through the SPRY4/p38 MAPK pathway.
Molecular mechanism: circPFKP functions as a cytoplasmic ceRNA sponge for miR-4516, thereby relieving miR-4516-mediated repression of SPRY4 and regulating p38 MAPK signaling.
Biological pathway or process:

ceRNA regulation (other); MAPK (inhibits); proliferation (inhibits); migration (inhibits); invasion (inhibits); apoptosis (inhibits); radioresistance (promotes)

Detected method:
Q
M
Validation methods:

Back-Splice Junction PCR / divergent primers PCR; Sanger Sequencing; RT-qPCR; Microarray; FISH / smFISH; Clinical Sample Validation; Bioinformatics Analysis; Luciferase Reporter Assay; Transfection; CCK8; Colony Formation Assay; Wound Healing Assay; Transwell Assay; Annexin V/PI Flow Cytometry; Western Blot; In Vivo Animal Model

Clinical significance:

circPFKP is significantly upregulated in PTC tissues and is highlighted as a potential novel therapeutic target for PTC patients.

Description:

circPFKP is an upregulated circRNA in PTC derived from PFKP exons 18 and 19. It mainly localizes to the cytoplasm and acts as a ceRNA sponge for miR-4516 to upregulate SPRY4, thereby modulating p38 MAPK signaling. Functionally, circPFKP suppresses proliferation, migration, invasion, and tumorigenicity under baseline conditions, but it also reduces apoptosis under stress or irradiation, suggesting a dual role and therapeutic relevance in PTC.

Confidence score:

0.7898

Other information
Title:

CircPFKP orchestrates a novel competing endogenous RNA network to regulate SPRY4/p38-MAPK signaling and modulate papillary thyroid carcinoma aggressiveness.

Journal: International journal of biological macromolecules
Published: 2025
PubMed ID: 41075905
Study type:

combined biological and clinical study

Data availability: GSE93522; GSE113629; GSE35570; TCGA; Supplementary Table 1; Supplementary Table 2; Supplementary Table 3; https://doi.org/10.1016/j.ijbiomac.2025.148158
Code availability: -