circRNA basic information
circBase ID: hsa_circ_0000199
Name: hsa_circ_AKT3
Synonym: circ_0000199 / circAKT3
Host Gene: AKT3
Genomic location(hg19): chr1:243708811-243736350:-
Genomic location(hg38): chr1:243545509-243573048:-
Subcellular localization: not tested
 
 
 
 
 
 
 
Disease basic information
MONDO ID:
0001056
MONDO name: gastric cancer
Disease details: gastric cancer / GC
Disease DO ID:
10534
Disease MeSH ID:
-
Disease NCIt ID:
C9331
Disease ICD11 ID:
1397617262
Disease OMIM ID:
613659
Species: Human
Species details: Homo sapiens
Tissue specimen:

tumor tissues; matched normal tissues

Cell lines:

MKN-7; HGC-27; GES-1; 293T

In vivo animal model:

cell line-derived xenograft

circRNA-disease information
Expression pattern:
UP
Associated gene: SLC1A5, Ago2
Associated microRNA: miR-515-5p
Biological function: circAKT3 promotes gastric cancer cell proliferation, survival, glutamine metabolism and tumor growth; circAKT3 knockdown inhibits proliferation, survival, glutamine uptake and in vivo tumor growth and promotes apoptosis.
Molecular mechanism: circAKT3 acts as a miR-515-5p sponge and relieves miR-515-5p-mediated inhibition of SLC1A5, thereby increasing SLC1A5 expression and promoting malignant behaviors and glutamine metabolism in gastric cancer cells.
Biological pathway or process:

proliferation (promotes); apoptosis (inhibits); glutaminolysis (promotes); ceRNA regulation (promotes)

Detected method:
Q
Validation methods:

RNase R Treatment; Actinomycin D / DRB Stability Assay; RT-qPCR; Clinical Sample Validation; Transfection; CCK8; EdU Staining; Colony Formation Assay; Annexin V/PI Flow Cytometry; Western Blot; Bioinformatics Analysis; Luciferase Reporter Assay; RIP (RNA Immunoprecipitation); IHC (Immunohistochemistry); In Vivo Animal Model

Clinical significance:

-

Description:

circAKT3 is up-regulated in gastric cancer tissues and cell lines. It functions as an oncogenic circRNA by sponging miR-515-5p to increase SLC1A5 expression, thereby promoting proliferation, survival, glutamine metabolism and tumor growth. Knockdown of circAKT3 suppresses malignant phenotypes and may represent a potential therapeutic strategy.

Confidence score:

0.8298

Other information
Title:

CircAKT3 promotes cell proliferation, survival and glutamine metabolism of gastric cancer by activating SLC1A5 expression via targeting miR-515-5p.

Journal: Histology and histopathology
Published: 2022
PubMed ID: 34850965
Study type:

combined biological and clinical study

Data availability: The datasets used and analyzed during the current study are available from the corresponding author on reasonable request.
Code availability: -