circRNA basic information
circBase ID: -
Name: hsa_circ_FGFR1
Synonym: circFGFR1int2
Host Gene: FGFR1
Genomic location(hg19): -
Genomic location(hg38): -
Subcellular localization: nucleus and cytoplasm
 
 
 
 
 
 
 
Disease basic information
MONDO ID:
0008315
MONDO name: prostate cancer
Disease details: prostate cancer / PCa
Disease DO ID:
10283
Disease MeSH ID:
D011471
Disease NCIt ID:
C7378
Disease ICD11 ID:
-
Disease OMIM ID:
-
Species: Human
Species details: Homo sapiens
Tissue specimen:

prostate adenocarcinomas tissue; benign prostatic hyperplasia (BPH) tissue; PCa tissue

Cell lines:

PC-3; DU145; LNCaP; 22Rv1; RWPE-1

In vivo animal model:

-

circRNA-disease information
Expression pattern:
UP
Associated gene: FGFR1, P65, FUS, AGO2, FGFR1 promoter
Associated microRNA: hsa-miR-4687-5p
Biological function: promotes PCa cell growth, migration, and invasion; promotes proliferation and DNA replication
Molecular mechanism: facilitates FGFR1 transcription by recruiting transcription activators P65/FUS and interacting with FGFR1 promoter; suppresses miR-4687-5p inhibitory effects on FGFR1 mRNA via competitive binding (miRNA sponge/ceRNA-like); co-exists with AGO2 in RISC
Biological pathway or process:

proliferation (promotes); migration (promotes); invasion (promotes); ceRNA regulation (promotes)

Detected method:
Q
H
Validation methods:

Back-Splice Junction PCR / divergent primers PCR; RNase R Treatment; Sanger Sequencing; RT-qPCR; ISH (In Situ Hybridization); Nuclear-Cytoplasmic Fractionation; Clinical Sample Validation; Bioinformatics Analysis; RIP (RNA Immunoprecipitation); RNA Pull-Down; ChIP / ChIP-seq; Luciferase Reporter Assay; Transfection; CCK8; EdU Staining; Transwell Assay; Wound Healing Assay; Cohort Study; Survival Analysis

Clinical significance:

Overexpression of circFGFR1int2 is significantly correlated with higher tumor grade, Gleason score, and PSA level, and is a significant unfavorable prognosticator for CRPC-free survival (CFS) (RR = 3.277, 95% confidence interval: 1.192-9.009; P = 0.021).

Description:

circFGFR1int2 is up-regulated in prostate cancer and promotes tumor cell proliferation, migration, and invasion. It enhances FGFR1 expression by recruiting P65/FUS to the FGFR1 promoter to activate transcription and by sponging miR-4687-5p to relieve post-transcriptional repression of FGFR1. High circFGFR1int2 level correlates with higher grade/Gleason score/PSA and predicts worse CRPC-free survival.

Confidence score:

0.8905

Other information
Title:

A novel intronic circular RNA circFGFR1int2 up-regulates FGFR1 by recruiting transcriptional activators P65/FUS and suppressing miR-4687-5p to promote prostate cancer progression.

Journal: Journal of translational medicine
Published: 2023
PubMed ID: 37993879
Study type:

combined biological and clinical study

Data availability: Data reported in the study shall be available upon reasonable request.
Code availability: -