circRNA basic information
circBase ID: -
Name: hsa_circ_ITCH
Synonym: circRNA itchy E3 ubiquitin protein ligase
Host Gene: ITCH
Genomic location(hg19): -
Genomic location(hg38): -
Subcellular localization: cytoplasm
 
 
 
 
 
 
 
Disease basic information
MONDO ID:
0009807
MONDO name: osteosarcoma
Disease details: osteosarcoma
Disease DO ID:
3347
Disease MeSH ID:
D012516
Disease NCIt ID:
C9145
Disease ICD11 ID:
-
Disease OMIM ID:
-
Species: Human
Species details: Homo sapiens
Tissue specimen:

OS tissue samples; matched non-tumor tissue samples; normal tissue samples

Cell lines:

hFOB 1.19; MG-63; KHOS; MG-63/DXR; KHOS/DXR

In vivo animal model:

cell line-derived xenograft

circRNA-disease information
Expression pattern:
DN
Associated gene: RASSF6
Associated microRNA: miR-524
Biological function: Overexpression of circITCH suppresses OS cell viability, migration and invasion, promotes apoptosis, reduces doxorubicin resistance, and constrains tumor growth in vivo.
Molecular mechanism: circITCH acts as a ceRNA sponge for miR-524 to up-regulate RASSF6, thereby repressing OS progression and reducing doxorubicin resistance.
Biological pathway or process:

proliferation (inhibits); migration (inhibits); invasion (inhibits); apoptosis (promotes); drug resistance (inhibits); chemoresistance (inhibits); ceRNA regulation (other)

Detected method:
Q
Validation methods:

RNase R Treatment; RT-qPCR; Nuclear-Cytoplasmic Fractionation; Clinical Sample Validation; Bioinformatics Analysis; Luciferase Reporter Assay; RIP (RNA Immunoprecipitation); Transfection; CCK8; Transwell Assay; Annexin V/PI Flow Cytometry; Western Blot; In Vivo Animal Model

Clinical significance:

circITCH was down-regulated in OS tissue samples and was lower in DXR-resistant patients than DXR-sensitive cases, suggesting relevance to OS development and doxorubicin resistance.

Description:

circITCH is down-regulated in osteosarcoma tissues, OS cell lines, and doxorubicin-resistant samples/cells. Its overexpression suppresses OS malignant phenotypes and doxorubicin resistance by sponging miR-524 to up-regulate RASSF6, and it also reduces xenograft tumor growth in vivo.

Confidence score:

0.7795

Other information
Title:

Down-regulation of circITCH promotes osteosarcoma development and resistance to doxorubicin via the miR-524/RASSF6 axis.

Journal: The journal of gene medicine
Published: 2021
PubMed ID: 34151476
Study type:

combined biological and clinical study

Data availability: The data and material presented in this manuscript are available from the corresponding author upon reasonable request.
Code availability: -