circRNA basic information
circBase ID: hsa_circ_0005941
Name: hsa_circ_FTO
Synonym: circFTO
Host Gene: FTO
Genomic location(hg19): chr16:53907697-53922863:+
Genomic location(hg38): chr16:53873785-53888951:+
Subcellular localization: cytoplasm
 
 
 
 
 
 
 
Disease basic information
MONDO ID:
0008383
MONDO name: rheumatoid arthritis
Disease details: Rheumatoid arthritis / RA
Disease DO ID:
7148
Disease MeSH ID:
D001172
Disease NCIt ID:
C2884
Disease ICD11 ID:
576319925
Disease OMIM ID:
180300
Species: Human
Species details: Homo sapiens
Tissue specimen:

synovial tissues; cartilage tissues

Cell lines:

HEK-293T

In vivo animal model:

other disease animal model

circRNA-disease information
Expression pattern:
UP
Associated gene: WTAP, METTL3, METTL14, SOX9, YTHDF2
Associated microRNA: -
Biological function: Promotes rheumatoid arthritis progression; inhibits chondrocyte proliferation, migration and anabolism; promotes chondrocyte apoptosis and catabolism; regulates chondrocyte metabolic balance.
Molecular mechanism: circFTO binds and facilitates assembly of the WTAP/METTL3/METTL14 m6A methyltransferase complex, increasing global m6A and enhancing m6A modification on SOX9 3’UTR, leading to reduced SOX9 mRNA stability; YTHDF2 mediates SOX9 mRNA degradation in an m6A-dependent manner.
Biological pathway or process:

m6A modification (promotes); mRNA stability (inhibits); apoptosis (promotes); proliferation (inhibits); migration (inhibits); other pathway/process (other)

Detected method:
Q
S
Validation methods:

RNA-seq; RT-qPCR; RNase R Treatment; Actinomycin D / DRB Stability Assay; FISH / smFISH; RNA Pull-Down; RIP (RNA Immunoprecipitation); Co-IP; Transfection; CCK8; Transwell Assay; TUNEL; Western Blot; In Vivo Animal Model; H&E Staining; Bioinformatics Analysis; Clinical Sample Validation

Clinical significance:

Increased expression of circFTO in synovial tissues from patients with RA; circFTO suggested as a therapeutic target for RA.

Description:

Exosomal circFTO derived from RA fibroblast-like synoviocytes is up-regulated in RA and aggravates disease by impairing chondrocyte proliferation/migration and anabolic activity while promoting apoptosis and catabolism. Mechanistically, circFTO interacts with and promotes assembly of the WTAP/METTL3/METTL14 m6A writer complex, increasing m6A on SOX9 mRNA and reducing SOX9 mRNA stability via YTHDF2-dependent decay. circFTO knockdown alleviates arthritis phenotypes in the CIA mouse model.

Confidence score:

0.8354

Other information
Title:

Fibroblast-like synoviocytes-derived exosomal circFTO deteriorates rheumatoid arthritis by enhancing N6-methyladenosine modification of SOX9 in chondrocytes.

Journal: Arthritis research & therapy
Published: 2024
PubMed ID: 38388473
Study type:

combined biological and clinical study

Data availability: available from the corresponding author upon reasonable request
Code availability: -