circRNA basic information
circBase ID: -
Name: hsa_circ_FAM114A2
Synonym: CircFAM114A2
Host Gene: FAM114A2
Genomic location(hg19): -
Genomic location(hg38): -
Subcellular localization: nucleus and cytoplasm
 
 
 
 
 
 
 
Disease basic information
MONDO ID:
0040679
MONDO name: urothelial carcinoma
Disease details: urothelial carcinoma
Disease DO ID:
-
Disease MeSH ID:
-
Disease NCIt ID:
C4030
Disease ICD11 ID:
-
Disease OMIM ID:
-
Species: Human
Species details: Homo sapiens
Tissue specimen:

urothelial carcinoma tumor tissues; adjacent normal tissues

Cell lines:

SV-HUC; BIU87; TCC; T24; RT4; 5637; 253J; UMUC3; J82; HEK293

In vivo animal model:

cell line-derived xenograft

circRNA-disease information
Expression pattern:
DN
Associated gene: P27, P21
Associated microRNA: miR-222-3p, miR-146a-5p
Biological function: Inhibits urothelial carcinoma cell proliferation, induces G1 cell cycle arrest and apoptosis, and increases cisplatin sensitivity/attenuates cisplatin chemoresistance.
Molecular mechanism: circFAM114A2 acts as a miRNA sponge for miR-222-3p and miR-146a-5p, thereby relieving repression of P27 and P21 (respectively) and promoting G1 arrest and cisplatin chemosensitivity.
Biological pathway or process:

cell cycle (inhibits); proliferation (inhibits); apoptosis (promotes); chemoresistance (inhibits); ceRNA regulation (other)

Detected method:
Q
S
Validation methods:

RNA-seq; RT-qPCR; RNase R Treatment; Sanger Sequencing; Back-Splice Junction PCR / divergent primers PCR; FISH / smFISH; Bioinformatics Analysis; RNA Pull-Down; Luciferase Reporter Assay; Transfection; CCK8; Cell Cycle Assay; Annexin V/PI Flow Cytometry; Colony Formation Assay; In Vivo Animal Model; Western Blot; IHC (Immunohistochemistry); Clinical Sample Validation; Cohort Study; Survival Analysis

Clinical significance:

Higher circFAM114A2 expression was associated with lower histological grade and better overall survival in urothelial carcinoma patients, suggesting prognostic biomarker potential.

Description:

circFAM114A2 is downregulated in urothelial carcinoma and functions as a tumor-suppressive circRNA. It sponges miR-222-3p and miR-146a-5p to upregulate P27 and P21, promoting G1 arrest and apoptosis and enhancing cisplatin sensitivity in vitro and in xenograft models; higher expression predicts better survival.

Confidence score:

0.8823

Other information
Title:

CircFAM114A2 Promotes Cisplatin Sensitivity via miR-222-3p/P27 and miR-146a-5p/P21 Cascades in Urothelial Carcinoma.

Journal: Frontiers in oncology
Published: 2021
PubMed ID: 34722233
Study type:

combined biological and clinical study

Data availability: https://www.frontiersin.org/articles/10.3389/fonc.2021.659166/full#supplementary-material
Code availability: -